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CAS: 2376137-31-2
Chemical Name: N1-(2-(((S)-2-(4-Chlorophenyl)-3-(4-((5R,7R)-7-hydroxy-5-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)piperazin-1-yl)-3-oxopropyl)amino)ethyl)-N12-((S)-1-((2S,4R)-4-hydroxy-2-(((S)-1-(4-(4-methylthiazol-5-yl)phenyl)ethyl)carbamoyl)pyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)dodecanediamide
Purity: >98% (HPLC)
Novel and potent AKT proteolysis targeting chimera (PROTAC) von Hippel-Lindau (VHL)-recruiting degrader
Ref: https://pubs.acs.org/doi/10.1021/acs.jmedchem.1c01476
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