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Glixx Laboratorie
CAS: 2059148-58-0
Chemical Name: 1-(5-(4-Fluoro-2-(2-(1,3,5-trimethyl-1H-pyrazol-4-yl)ethoxy)phenyl)-1-methyl-1H-indazol-3-yl)-N,N-dimethylmethanamine
Purity: >98% (HPLC)
Novel resistance breaking antimalarial N-myristoyltransferase (NMT) inhibitor, binding to NMT peptide binding pocket
References:
1) https://journals.plos.org/plosbiology/article?id=10.1371/journal.pbio.3001408
2) https://www.sciencedirect.com/science/article/pii/S2451945619301114
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