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CAS: 2641993-55-5
Chemical Name: (3S)-N-((2S)-1-(((63S,4S)-11-Ethyl-12-(2-((S)-1-methoxyethyl)pyridin-3-yl)-10,10-dimethyl-5,7-dioxo-61,62,63,64,65,66-hexahydro-11H-8-oxa-1(5,3)-indola-6(1,3)-pyridazina-2(1,3)-benzenacycloundecaphane-4-yl)amino)-3-methyl-1-oxobutan-2-yl)-N-methyl-1-(4-morpholinobut-2-ynoyl)pyrrolidine-3-carboxamide
Purity: >98% (HPLC)
Novel, functionally distinct tricomplex KRASG12C active-state inhibitor, retaining the ability to bind and inhibiting KRASG12C/Y96D and overcoming resistance
Ref: https://cancerdiscovery.aacrjournals.org/content/early/2021/06/16/2159-8290.CD-21-0365.long
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