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CAS: N/A
Chemical Name: (2S,4R)-1-((2S)-2-(2-(2,2-bis-((R)-2-(2-(2-(2-(4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a]azepin-6-yl)acetamido)ethoxy)ethoxy)ethoxymethyl)propoxy)acetamido)-3,3-dimethylbutanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide
Purity: >98% (HPLC)
Novel trivalent PROTAC, acting as a low picomolar BET degrader with preference for bromodomain containing 2 (BRD2)
Ref: https://www.nature.com/articles/s41589-021-00878-4#Sec83
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