Glixx Laboratories Inc

               Your exclusive source for bioactive molecules

Glixx Laboratorie

 

   sales@glixxlabs.com      Toll-Free: (855)Go-Glixx   Tel: 781-333-5348    Fax: 781-333-5368 
SIM1

 

CAS: N/A

 

Chemical Name: (2S,4R)-1-((2S)-2-(2-(2,2-bis-((R)-2-(2-(2-(2-(4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a]azepin-6-yl)acetamido)ethoxy)ethoxy)ethoxymethyl)propoxy)acetamido)-3,3-dimethylbutanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide

 

 
GLXC-24725For Lab R&D Uses Only
        Cat No: GLXC-24725

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel trivalent PROTAC, acting as a low picomolar BET degrader with preference for bromodomain containing 2 (BRD2)

 

Ref: https://www.nature.com/articles/s41589-021-00878-4#Sec83

 

Analytical data click for PDF file

 

 

Place an order!

Price & Availability





POA
 








Bulk inquiry contact:
sales@glixxlabs.com
service@glixxlabs.com