Glixx Laboratories Inc

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MS83

 

CAS: 2762181-19-9

 

Chemical Name: Ethyl (S)-3-(7-(2-(2-(2-((S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)acetamido)acetamido)ethoxy)-1-methyl-1H-benzo[d][1,2,3]triazol-5-yl)-3-(4-methyl-3-(((R)-4-methyl-1,1-dioxido-3,4-dihydro-2H-benzo[b][1,4,5]oxathiazepin-2-yl)methyl)phenyl)propanoate

 

 
GLXC-26971For Lab R&D Uses Only
        Cat No: GLXC-26971

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel BRD4/3 degrader, effectively reducing protein levels of BRD4 and BRD3, but not BRD2, in cells in a concentration-, time-, KEAP1- and UPS-dependent manner, degrading BRD4/3 more durably than the CRBN-recruiting PROTAC dBET1 in MDA-MB-468 cells and selectively degrading BRD4 short isoform over long isoform in MDA-MB-231 cells

 

Reference:

https://www.ncbi.nlm.nih.gov/pmc/articles/PMC8480205/

 

Analytical data click for PDF file

 

 

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