Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 1426214-64-3
Chemical Name: Sgk1-IN-2; N-(4-(3-Amino-1H-pyrazolo[3,4-b]pyrazin-6-yl)phenyl)-2,5-dichlorobenzenesulfonamide
Purity: >98% (HPLC)
Novel potent inhibitor of SGK1/3, reducing PI3K-Akt inhibitor resistant cell growth, possessing an IC50 of 4 nM for SGK3, 10 nM for SGK1, and 76 nM for S6K1
References:
1) https://pdfs.semanticscholar.org/2559/77367dfa429f101f6420324779365c7c881c.pdf
2) https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4291729/
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