Glixx Laboratories Inc

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Glixx Laboratorie

 

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UM-203

 

CAS: N/A

 

Chemical Name: N-(1-(2-Ethynylthiazole-4-carbonyl)-4-(1-methyl-1H-benzo[d]imidazol-2-yl)piperidin-4-yl)-2-phenylthiazole-5-carboxamide

 

 
GLXC-90186For Lab R&D Uses Only
        Cat No: GLXC-90186

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel reversible covalent STING antagonist, maintaining activity against the most prevalent human STING variant (R232), effectively suppressing STING signaling in primary human CD14+ monocytes, and exhibiting moderate metabolic stability

 

Reference:

https://pubs.acs.org/doi/10.1021/acsmedchemlett.5c00611

 

Analytical data click for PDF file

 

 

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