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CAS: 2503017-97-6
Chemical Name: 3-(4-(10-(((S)-2-(4-Chlorophenyl)-3-(4-((5R,7R)-7-hydroxy-5-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)piperazin-1-yl)-3-oxopropyl)amino)decyl)-1-oxoisoindolin-2-yl)piperidine-2,6-dione
Purity: >98% (HPLC)
Novel selective pan-AKT degrader, inducing potent degradation of all three AKT isoforms and displaying enhanced anti-proliferative effects relative to GDC-0068, promoting sustained AKT degradation and inhibition of downstream signaling effects for up to 96 h
Refernces:
1) https://www.sciencedirect.com/science/article/abs/pii/S2451945619303964
2) https://www.biorxiv.org/content/10.1101/848887v1.full
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