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CAS: 2140807-05-0
Chemical Name: 2-(5-Fluoro-2-hydroxyphenyl)-2-(1-oxo-6-(4-(piperazin-1-yl)phenyl)isoindolin-2-yl)-N-(thiazol-2-yl)acetamide
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel mutant-selective EGFR allosteric inhibitor, inhibiting cell proliferation and EGFRL858R/T790M/C797S signaling in vitro and in vivo
Reference:
https://cancerdiscovery.aacrjournals.org/content/9/7/926.long
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