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Antiallergic Agent 36

 

CAS: N/A

 

Chemical Name: 3-((2-Amino-5-(1-methyl-1H-pyrazol-4-yl)pyridin-3-yl)ethynyl)-N-(3,5-bis(trifluoromethyl)phenyl)-4-methylbenzamide

 

 
GLXC-24446For Lab R&D Uses Only
        Cat No: GLXC-24446

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel highly potent orally bioavailable antiallergic agent, effectively suppressing mast cell degranulation in a dose-dependent manner (IC50, 2.54 nM for RBL-2H3 cells; 48.28 nM for peritoneal mast cells (PMCs))

 

Ref: https://pubs.acs.org/doi/10.1021/acs.jmedchem.1c00976

 

Analytical data click for PDF file

 

 

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