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CAS: N/A
Chemical Name: LGR4455; 5-((2-Aminoethyl)thio)-3-isopropyl-N-(4-(pyridin-2-yl)benzyl)-2H-pyrazolo[4,3-d]pyrimidin-7-amine
Purity: >98% (HPLC)
Novel potent inhibitor of cyclin-dependent kinases (CDKs) 2, 5, and 9, displaying activities across more than 60 cancer cell lines
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.9b00189
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