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CAS: N/A
Chemical Name: 3-Hydroxy-2-methyl-1-(8-(4-(4-((2-(pyrrolidin-1-ylmethyl)-1H-benzo[d]imidazol-1-yl)methyl)phenyl)-1H-1,2,3-triazol-1-yl)octyl)pyridin-4(1H)-one
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel potent histone lysine demethylase inhibitor (KDMi), causing transcriptome-level perturbations favoring cell cycle inhibition and apoptosis
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.5c02018
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